29 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Article Title
Organization
Development of Glucose Regulated Protein 94-Selective Inhibitors Based on the BnIm and Radamide Scaffold.
The University of Kansas
Structure-Activity Relationships of the Peptide Kappa Opioid Receptor Antagonist Zyklophin.
The University of Kansas
Studies toward the Development of Antiproliferative Neoclerodanes from Salvinorin A.
The University of Kansas
Synthesis and¿-opioid receptor activity of furan-substituted salvinorin A analogues.
The University of Kansas
Are MDCK cells transfected with the human MRP2 gene a good model of the human intestinal mucosa?
The University of Kansas
Are MDCK cells transfected with the human MDR1 gene a good model of the human intestinal mucosa?
The University of Kansas
The sulfonimidamide as a novel transition state analog for aspartic acid and metallo proteases.
The University of Kansas
Discovery of dermorphin-based affinity labels with subnanomolar affinity for mu opioid receptors.
The University of Kansas
Design, synthesis, and pharmacological activities of dynorphin A analogues cyclized by ring-closing metathesis.
The University of Kansas
Synthesis of 4,5,6,7-tetrahydrothieno[3,2-c]pyridines and comparison with their isosteric 1,2,3,4-tetrahydroisoquinolines as inhibitors of phenylethanolamine N-methyltransferase.
The University of Kansas
Synthesis and pharmacological characterization of novel fluorescent histamine H2-receptor ligands derived from aminopotentidine.
The University of Kansas
Design, synthesis, and biological evaluation of aminoalkylindole derivatives as cannabinoid receptor ligands with potential for treatment of alcohol abuse.
The University of Kansas
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
The University of Kansas
Isolation and characterization of Caco-2 subclones expressing high levels of multidrug resistance protein efflux transporter.
The University of Kansas
A functional assay for quantitation of the apparent affinities of ligands of P-glycoprotein in Caco-2 cells.
The University of Kansas
Click chemistry to probe Hsp90: Synthesis and evaluation of a series of triazole-containing novobiocin analogues.
The University of Kansas
Synthesis and evaluation of Hsp90 inhibitors that contain the 1,4-naphthoquinone scaffold.
The University of Kansas
Addressing Structural Flexibility at the A-Ring on Salvinorin A: Discovery of a Potent Kappa-Opioid Agonist with Enhanced Metabolic Stability.
The University of Kansas
Transformation of the Non-Selective Aminocyclohexanol-Based Hsp90 Inhibitor into a Grp94-Seletive Scaffold.
The University of Kansas